- Isolation, structure determination, and synthesis of galaxamide, a rare cytotoxic cyclic pentapeptide from a marine algae Galaxaura filamentosa.
[作者:Xu, Wen-Jie;Liao, Xiao-Jian;Xu, Shi-Hai;Diao, Jian-Zhong;Du, Bin;Zhou, Xu-Long;Pan, Shan-Shan;,期刊:Organic Letters, 页码:4569-4572 , 文章类型: 研究论文,,卷期:2008年10-20]
- Galaxamide (I), cyclo(-N-MeLeu-Leu-N-MeLeu-Leu-Leu-), a rare cyclic pentapeptide, was isolated from G. filamentosa. A preliminary bioassay of I showed marked in vitro antiproliferative activities against GRC-1 and HepG2...
- Synthesis of anthracene and azaanthracene fluorophores via [2+2+2] cyclotrimerization reactions.
[作者:Zou, Yan;Young, Douglas D.;Cruz-Montanez, Alejandra;Deiters, Alexander;,期刊:Organic Letters, 页码:4661-4664 , 文章类型: 研究论文,,卷期:2008年10-20]
- Organic Pigments, Fluorescent Brighteners, and Photographic A highly convergent [2+2+2] cyclotrimerization approach to anthracenes and 2-azaanthracenes has been developed. It allows for the facile introduction of the an...
- A new total synthesis of patellamide A.
[作者:Garcia-Reynaga, Pablo;VanNieuwenhze, Michael S.;,期刊:Organic Letters, 页码:4621-4623 , 文章类型: 研究论文,,卷期:2008年10-20]
- Patellamide A, cytotoxic and antitumor lipophilic cyclic peptide isolated from marine tunicate Lissoclinum patella, was efficiently synthesized from thiazole (I) (Fmoc = 9-fluorenyl methoxy carbonyl) via two complementar...
- A Tandem One-Pot, Microwave-Assisted Synthesis of Regiochemically Differentiated 1,2,4,5-Tetrahydro-1,4-benzodiazepin-3-ones.
[作者:De Silva, Ravindra A.;Santra, Soumava;Andreana, Peter R.;,期刊:Organic Letters, 页码:4541-4544 , 文章类型: 研究论文,,卷期:2008年10-20]
- A one-pot, two-step synthesis of the title compds. employs a multicomponent Ugi condensation reaction, microwave irradn., and Fe(0) as a reductant. Two pathways are accessible; both routes utilize bifunctional, o-nitro-...
- Enantiopure 2-Substituted Glyceraldehyde Derivatives by Aza-Claisen Rearrangement or C-Alkylation of Enamines.
[作者:Bridgwood, Katy L.;Tzschucke, C. Christoph;O'Brien, Matthew;Wittrock, Sven;Goodman, Jonathan M.;Davies, John E.;Logan, Angus W. J.;Huttl, Matthias R. M.;Ley, Steven V.;,期刊:Organic Letters, 页码:4537-4540 , 文章类型: 研究论文,,卷期:2008年10-20]
- 2-Alkyl derivs. of butane-2,3-diacetal-protected glyceraldehyde I (R1 = Me, NCCH2, HCYCCH2, H2C:CHCH2, EtO2CCH2, PhCH2, etc.) were stereoselectively prepd. by aza-Claisen rearrangement of N-allyl-enammonium ions or C-alk...
- 1-Substituted 5-Aminotetrazoles: Syntheses from CNN3 with Primary Amines.
[作者:Joo, Young-Hyuk;Shreeve, Jean'ne M.;,期刊:Organic Letters, 页码:4665-4667 , 文章类型: 研究论文,,卷期:2008年10-20]
- 1-Substituted 5-aminotetrazoles, e.g., I, were prepd. in situ by an excellent reaction of cyanogen azide and primary amines to generate an imidoyl azide as an intermediate in acetonitrile/water. After cyclization, the i...
- A Formal Total Synthesis of Platencin.
[作者:Austin, Kerrie A. B.;Banwell, Martin G.;Willis, Anthony C.;,期刊:Organic Letters, 页码:4465-4468 , 文章类型: 研究论文,,卷期:2008年10-20]
- The readily available and enantiomerically pure trienes I undergo a thermally induced intramol. Diels-Alder reaction to give the corresponding mixt. of compds. II (R = OSiMe2CMe3, R1 = H; R = H, R1 = OSiMe2CMe3). This m...
- A Bench-Stable Pd Catalyst for the Hydroarylation of Fullerene with Boronic Acids.
[作者:Mori, Susumu;Nambo, Masakazu;Chi, Liang-Chen;Bouffard, Jean;Itami, Kenichiro;,期刊:Organic Letters, 页码:4609-4612 , 文章类型: 研究论文,,卷期:2008年10-20]
- A Pd(II) catalyst for the hydroarylation of fullerene with boronic acids is presented. Treatment of C60 with an arylboronic acid ArB(OH)2 (Ar = Ph, 4-MeC6H4, 4-ClC6H4, 4-AcC6H4, 3-thienyl, etc.) in the presence of a cat...
- Zirconocene-Mediated Synthesis of Cyclobutabenzenes.
[作者:Barluenga, Jose;Calleja, Jonas;Anton, Maria J.;Alvarez-Rodrigo, Lucia;Rodriguez, Felix;Fananas, Francisco J.;,期刊:Organic Letters, 页码:4469-4471 , 文章类型: 研究论文,,卷期:2008年10-20]
- A new, mild, one-pot method for the synthesis of cyclobutabenzenes, e.g., I, by the zirconium-promoted cross-coupling reaction of aryllithium compds. and alkenyl bromides is reported. Formation of an arynezirconocene co...
- Facile Preparation of a-Aryl Nitriles by Direct Cyanation of Alcohols with TMSCN Under the Catalysis of InX3.
[作者:Chen, Gang;Wang, Zheng;Wu, Jiang;Ding, Kuiling;,期刊:Organic Letters, 页码:4573-4576 , 文章类型: 研究论文,,卷期:2008年10-20]
- 23 A convenient and efficient synthesis of a-aryl nitriles, e.g., I, was developed by direct cyanation of alcs. with TMSCN under the catalysis of Lewis acid. Using 5-10 mol % of InBr3 as the catalyst, a variety of benzy...
|