- Efficient Synthesis of 4,7-Diamino Substituted 1,10-Phenanthroline-2,9-dicarboxamides
[作者:LARSEN ANDERS FOLLER; ULVEN TROND,期刊:Organic Letters, 页码:3546-3548 , 文章类型: Article,,卷期:2011年13-13]
- A convenient and high-yielding multigram synthesis of the versatile intermediate 4,7-dichloro-1,10-phenanthroline-2,9-dicarboxylic acid is described. The intermediate is further efficiently derivatized to 4,7-diamino-1,1...
- Asymmetric Synthesis of (+)-Mequitazine from Quinine
[作者:LEROUX SEBASTIEN; LARQUETOUX LAURENT; NICOLAS MARC; DORIS ERIC,期刊:Organic Letters, 页码:3549-3551 , 文章类型: Article,,卷期:2011年13-13]
- The first asymmetric synthesis of the antihistaminic drug mequitazine is reported. Our approach started from quinine, a Cinchona alkaloid, whose chiral information was exploited for setting up the stereogenic center of (...
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