- Targeting GSK3 from Ustilago maydis: Type-II Kinase Inhibitors as Potential Antifungals
[作者:GRUETTER CHRISTIAN; SIMARD JEFFREY R; MAYERWRANGOWSKI SVENJA C; SCHREIER PETER H; PEREZMARTIN JOSE; RICHTERS ANDRE; GETLIK MATTHAEUS; GUTBROD OLIVER; BRAUN CHRISTOPH A; BECK MICHAEL E; RAUH DANIEL,期刊:ACS CHEMICAL BIOLOGY, 页码:1257-1267 , 文章类型: Article,,卷期:2012年7-7]
- Protein kinases are key enzymes in the complex regulation of cellular processes in almost all living organisms. For this reason, protein kinases represent attractive targets to stop the growth of eukaryotic pathogens suc...
- A High-Throughput Screen To Identify Inhibitors of ATP Homeostasis in Non-replicating Mycobacterium tuberculosis
[作者:MAK PUIYING A; RAO SRINIVASA P S; TAN MAI PING; LIN XIUHUA; CHYBA JASON; TAY JOANN; NG SEOW HWEE; TAN BEE HUAT; CHERIAN JOSEPH; DURAISWAMY JEYARAJ; BIFANI PABLO; LIM VIVIAN; LEE BOON HENG; MA NGAI LING; BEER DAVID; THAYALAN PAMELA; KUHEN KELLI; CHATTERJEE ARNAB; SUPEK FRANTISEK; GLYNNE RICHARD; ZHENG JUN; BOSHOFF HELENA I; BARRY CLIFTON E III; DICK THOMAS; PETHE KEVIN; CAMACHO LUIS R,期刊:ACS CHEMICAL BIOLOGY, 页码:1190-1197 , 文章类型: Article,,卷期:2012年7-7]
- Growing evidence suggests that the presence of a subpopulation of hypoxic non-replicating, phenotypically drug-tolerant mycobacteria is responsible for the prolonged duration of tuberculosis treatment. The discovery of n...
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