- A Practical Synthesis of (-)-Kainic Acid
[作者:TAKITA SATOSHI; YOKOSHIMA SATOSHI; FUKUYAMA TOHRU,期刊:Organic Letters, 页码:2068-2070 , 文章类型: Article,,卷期:2011年13-8]
- A highly practical stereoselective total synthesis of (-)-kainic acid is described. This synthesis features the stereoselective alkylation of an iodolactone intermediate that was efficiently prepared from (+)-carvone and...
- Rapid One-Pot, Four-Step Synthesis of Highly Fluorescent 1,3,4,5-Tetrasubstituted Pyrazoles
[作者:WILLY BENJAMIN; MUELLER THOMAS J J,期刊:Organic Letters, 页码:2082-2085 , 文章类型: Article,,卷期:2011年13-8]
- 1,3,4,5-Tetrasubstituted pyrazoles can be rapidly and efficiently synthesized in a one-pot, four-step sequence consisting of Sonogashira coupling, addition-cyclocondensation, bromination, and Suzuki coupling. The second ...
- Regiocontrolled Rearrangement of Isobenzofurans
[作者:EGAN BEN A; PARADOWSKI MICHAEL; THOMAS LYNNE H; MARQUEZ RODOLFO,期刊:Organic Letters, 页码:2086-2089 , 文章类型: Article,,卷期:2011年13-8]
- The regioselective alkylation and oxidative rearrangement of isobenzofurans has been achieved to generate substituted 4,8-dihydroxyisochromanones in good yields and with complete regiocontrol.
- Total Synthesis and Biological Evaluation of (-)-9-Deoxy-englerin A
[作者:USHAKOV DMITRY B; NAVICKAS VAIDOTAS; STROEBELE MARKUS; MAICHLEMOESSMER CAECILIA; SASSE FLORENZ; MAIER MARTIN E,期刊:Organic Letters, 页码:2090-2093 , 文章类型: Article,,卷期:2011年13-8]
- An effective total synthesis of (-)-9-deoxy-englerin (4), an analogue of the natural guaiane sesquiterpene englerin A (1), has been achieved. The synthesis features a transannular epoxide opening to construct the 5,7-fus...
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