- Synthesis and Biological Evaluation of a New Series of 1,2,4-Triazolo[1,5-a]-1,3,5-triazines as Human A(2A) Adenosine Receptor Antagonists with Improved Water Solubility
[作者:FEDERICO STEPHANIE; PAOLETTA SILVIA; CHEONG SIEW LEE; PASTORIN GIORGIA; CACCIARI BARBARA; STRAGLIOTTO STEFANO; KLOTZ KARL NORBERT; SIEGEL JEFFREY; GAO ZHANGUO; JACOBSON KENNETH A; MORO STEFANO; SPALLUTO GIAMPIERO,期刊:Journal of Medicinal Chemistry, 页码:877-889 , 文章类型: Article,,卷期:2011年54-3]
- The structure-activity relationship (SAR) of 1,2,4-triazolo[1,5-a]-1,3,5-triazine derivatives related to ZM241385 as antagonists of the A(2A) adenosine receptor (AR) was explored through the synthesis of analogues substi...
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