- Discovery of a Highly Potent and Selective MEK Inhibitor: GSK1120212 (JTP-74057 DMSO Solvate)
[作者:ABE HIROYUKI; KIKUCHI SHINICHI; HAYAKAWA KAZUHIDE; IIDA TETSUYA; NAGAHASHI NOBORU; MAEDA KATSUYA; SAKAMOTO JOHEI; MATSUMOTO NORIAKI; MIURA TOMOYA; MATSUMURA KOJI; SEKI NORIYOSHI; INABA TAKASHI; KAWASAKI HISASHI; YAMAGUCHI TAKAYUKI; KAKEFUDA REINA; NANAYAMA TOYOMICHI; KURACHI HIRONORI; HORI YOSHIKAZU; YOSHIDA TAKAYUKI; KAKEGAWA JUNYA; WATANABE YOSHIHIRO; GILMARTIN AIDAN G; RICHTER MARK C; MOSS KATHERINE G; LAQUERRE SYLVIE G,期刊:ACS Medicinal Chemistry Letters, 页码:320-324 , 文章类型: Article,,卷期:2011年2-4]
- Inhibition of mitogen-activated protein kinase/extracellular signal-regulated kinase kinase (MEK) represents a promising strategy for the discovery of a new generation of anticancer chemotherapeutics. Our synthetic effor...
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