- Identification of a New Series of STAT3 Inhibitors by Virtual Screening
[作者:MATSUNO KENJI; MASUDA YOSHIAKI; UEHARA YUTAKA; SATO HIROSHI; MUROYA AYUMU; TAKAHASHI OSAMU; YOKOTAGAWA TAKANE; FURUYA TOSHIO; OKAWARA TADASHI; OTSUKA MASAMI; OGO NAOHISA; ASHIZAWA TADASHI; OSHITA CHIE; TAI SACHIKO; ISHII HIDEE; AKIYAMA YASUTO; ASAI AKIRA,期刊:ACS Medicinal Chemistry Letters, 页码:371-375 , 文章类型: Article,,卷期:2010年1-8]
- The signal transducer and activator of transcription 3 (STAT3) is considered to be an attractive therapeutic target for oncology drug development. We identified a N-[2-(1,3,4-oxadiazolyl)]-4-quinolinecarboxamide derivati...
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