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Design, synthesis and analgesic properties of novel conformationally-restricted N-acylhydrazones (NAH)

  作者 Kummerle, AE; Vieira, MM; Schmitt, M; Miranda, ALP; Fraga, CAM; Bourguignon, JJ; Barreiro, EJ  
  选自 期刊  Bioorganic & Medicinal Chemistry Letters;  卷期  2009年19-17;  页码  4963-4966  
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[摘要]A set of six azaheterocycles were designed as conformationnaly-constrained N-acylhydrazones and tested as analgesics. (C) 2009 Elsevier Ltd. All rights reserved.

 
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