EFFICIENT SYNTHESIS OF 5-AMINO-6-DIALKYLAMINO-4-HYDROXYPENTANAMIDE DERIVATIVES FOR RENIN INHIBITORS

[摘要]：We report an efficient synthetic method for 5-amino-6-dialkylamino-4-hydroxypentanamide derivatives using Shi Asymmetric Epoxidation and the ring opening of N-(2-nitrobenzenesulfonyl)aziridine with hindered secondary amine as key steps.

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