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Synthesis and biological evaluation of technetium-labeled D-glucose-MAG(3) derivative as agent for tumor diagnosis

  作者 de Barros, ALB; Cardoso, VN; Mota, LD; Leite, EA; de Oliveira, MC; Alves, RJ  
  选自 期刊  Bioorganic & Medicinal Chemistry Letters;  卷期  2009年19-9;  页码  2497-2499  
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[摘要]A D-glucose-MAG3 derivative was successfully synthesized and radiolabeled in high labeling yield. Biodistribution studies in Ehrlich tumor-bearing mice were performed. This compound showed high accumulation in tumor tissue with high tumor-to-muscle ratio and moderate tumor-to-blood ratio. Thus, Dglucose-MAG(3) is a potential agent for tumor diagnosis. (C) 2009 Elsevier Ltd. All rights reserved.

 
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