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[摘要]:An efficient, one-pot, multicomponent reaction of aldehydes 1, p-methoxyaniline (2a), and 2-vinylindoles 3 was developed. This approach provides a practical approach to synthetically and biologically significant tetrahydro-gamma-carboline and tetrahydroquinoline derivatives in good yields through a chemo-and regioselectivity switch, which can be tuned by simply changing the substituent on the indole component under identical reaction conditions. |
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