A FACILE SYNTHESIS OF 5,6-DIHYDRO-4H-PYRROLO[3,4-d]THIAZOLE AND OTHER PYRROLIDINE-FUSED AROMATIC RING SYSTEMS VIA ONE-STEP CYCLIZATION FROM DIOLS

[摘要]：A facile synthetic method of 5,6-dihydro-4H-pyrrolo[3,4-d]thiazole, which is a subunit of a potent factor Xa (fXa) inhibitor was developed. This new approach employs one-step cyclization from a diol and can be applied to the syntheses of other pyrrolidine-fused aromatic ring sytems.

[全文传递流程]：

一般上传文献全文的时限在1个工作日内