AN IMPROVED SYNTHESIS OF ARYLBORONATES TOWARD TWENTY NOVEL 1,3-DISUBSTITUTED 4-AMINO-1H-PYRAZOLO[3,4-d]PYRIMIDINE ANALOGS
[摘要]:By developing an improved procedure for arylboronates, twenty 1H-pyrazolo[3,4-d]pyrimidine analogs were efficiently synthesized as a source of a potent kinase inhibitor.
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