- A New Mild Method for the C-Acylation of Ketone Enolates. A Convenient Synthesis of beta-Keto-Esters, -Thionoesters, and -Thioesters
[作者:HALE KARL J; GRABSKI MILOSZ; FLASZ JAKUB T,期刊:Organic Letters, 页码:370-373 , 文章类型: Article,,卷期:2013年15-2]
- A new method for ketone enolate C-acylation is described which utilizes alkyl pentafluorophenylcarbonates, thiocarbonates, and thionocarbonates as the reactive acylating agents, and MgBr2 center dot Et2O, DMAP, and i-Pr2...
- Addition of Cyclic Ureas and 1-Methyl-2-oxazolidone to Pyridynes: A New Approach to Pyridodiazepines, Pyridodiazocines, and Pyridooxazepines
[作者:SAITO NOZOMI; NAKAMURA KENICHI; SHIBANO SAYAKO; IDE SOICHIRO; MINAMI MASABUMI; SATO YOSHIHIRO,期刊:Organic Letters, 页码:386-389 , 文章类型: Article,,卷期:2013年15-2]
- Reactions of pyridynes with cyclic urea and 1-methyl-2-oxazolidone were demonstrated. 3,4-Pyridyne and 2,3-pyridyne were reacted with N,N-dimethylimidazolidone, N,N-dimethylpropylene urea, and 1-methyl-2-oxazolidone to g...
- Hunanamycin A, an Antibiotic from a Marine-Derived Bacillus hunanensis
[作者:HU YOUCAI; WANG KEZHAN; MACMILLAN JOHN B,期刊:Organic Letters, 页码:390-393 , 文章类型: Article,,卷期:2013年15-2]
- Hunanamycin A, the first natural product with a pyrido[1,2,3-de]quinoxaline-2,3-dione core, was isolated from a marine-derived Bacillus hunanensis. Hunanamycin A is related to a degradation product of riboflavin but has ...
- Stereocontrolled Synthesis of the AB Rings of Samaderine C
[作者:BURNS DAVID J; MOMMER STEFAN; OBRIEN PETER; TAYLOR RICHARD J K; WHITWOOD ADRIAN C; HACHISU SHUJI,期刊:Organic Letters, 页码:394-397 , 文章类型: Article,,卷期:2013年15-2]
- A concise synthesis of the AB rings of samaderine C (12 steps, 8 isolation steps, 7.8% overall yield), a quassinoid with antifeedant and insecticidal activity, is described. The development of the first general approach ...
- Total Synthesis of Kingianin A
[作者:LIM HEE NAM; PARKER KATHLYN A,期刊:Organic Letters, 页码:398-401 , 文章类型: Article,,卷期:2013年15-2]
- A 12-step synthesis of kingianin A, an inhibitor of the antiapoptotic protein Bcl-xL, Is based on a radical cation Diels-Alder reaction (RCDA). This approach is thought to be biomimetic. The use of a tether in the key RC...
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