- Cyclic Peptide Synthesis with Thioacids
[作者:SASAKI KANAME; CRICH DAVID,期刊:Organic Letters, 页码:3254-3257 , 文章类型: Article,,卷期:2010年12-14]
- C-Terminal amino acid 9-fluorenylmethylthioesters may be carried through Boc chemistry solution phase peptide synthesis sequences. After insertion of the final residue in the form of an Fmoc carbamate, treatment with pip...
- A New Synthesis of 2,3-Di- or 2,3,3-Trisubstituted 2,3-Dihydro-4-pyridones by Reaction of 3-Ethoxycyclobutanones and N-p-Toluenesulfonyl Imines Using Titanium(IV) Chloride: Synthesis of (+/-)-Bremazocine
[作者:MATSUO JUNICHI; OKADO RYOHEI; ISHIBASHI HIROYUKI,期刊:Organic Letters, 页码:3266-3268 , 文章类型: Article,,卷期:2010年12-14]
- N-p-Toluenesulfonyl (Ts) aldimines reacted with 3-ethoxycyclobutanones by catalysis of titanium(IV) chloride to afford 2,3-di- or 2,3,3-trisubstituted N-Ts-2,3-dihydro-4-pyridones. Synthesis of (+/-)-bremazocine was effi...
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