- Polymer-Supported Stereoselective Synthesis of Benzimidazolinopiperazinones
[作者:CANKAROVA NADEZDA; KRCHNAK VIKTOR,期刊:Journal of Organic Chemistry, 页码:5687-5695 , 文章类型: Article,,卷期:2012年77-13]
- We describe the efficient synthesis of 4,7,8,10-tetrasubstituted-((( 4S 10aS)-3-oxo -3,4,10,10a-tetrahydrobenzo[4,5]imidazo[1,2-a]pyrazin-2(1H)-yl)alkyl)amides on solid phase via tandem N-acyliminium ion cyclization-nucl...
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