- Palladium-Catalyzed 2-Arylation of Pyrroles
[作者:GRYKO DANIEL T; VAKULIUK OLENA; GRYKO DOROTA; KOSZARNA BEATA,期刊:Journal of Organic Chemistry, 页码:9517-9520 , 文章类型: Article,,卷期:2009年74-24]
- A methodology that affords N-alkyl-2-arylpyrroles and N-aryl-2-arylpyrroles via direct coupling from aryl iodides has been developed. After examining various reaction parameters: solvent, ratio of reagents, catalyst, bas...
- Reduction of Solid-Supported Olefins and Alkynes
[作者:DICKSON DAVID P; TOH CHRISTINE; LUNDA MENAKA; YERMOLINA MARIA V; WARDROP DUNCAN J; LANDRIE CHAD L,期刊:Journal of Organic Chemistry, 页码:9535-9538 , 文章类型: Article,,卷期:2009年74-24]
- The reduction of carbon-carbon multiple bonds in alkynes and olefins supported on a polystyrene resin has been investigated. Homogeneous catalysis by titanocene reagents is effective for the stereoselective preparation o...
- Synthesis of a TRPV1 Receptor Antagonist
[作者:YU SU; HAIGHT ANTHONY; KOTECKI BRIAN; WANG LEI; LUKIN KIRILL; HILL DAVID R,期刊:Journal of Organic Chemistry, 页码:9539-9542 , 文章类型: Article,,卷期:2009年74-24]
- A five-step synthesis of a TRPV1 receptor antagonist 1 is described. The key step involves a novel palladium-catalyzed amidation reaction of 4-chloro-1-methylindazole 8 with the benzyl urea 9 to form the unsymmetrically ...
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