- Total Synthesis of Lodopyridone
[作者:BURCKHARDT TOBIAS; HARMS KLAUS; KOERT ULRICH,期刊:Organic Letters, 页码:4674-4677 , 文章类型: Article,,卷期:2012年14-17]
- A convergent total synthesis of the structurally unprecedented alkaloid lodopyridone was achieved using a cross-coupling of an lodopyridone fragment with a quinolinethiazolylstannane. Key features of the syntheses of the...
- Total Synthesis of Pentosidine
[作者:ROSENBERG ADAM J; CLARK DANIEL A,期刊:Organic Letters, 页码:4678-4681 , 文章类型: Article,,卷期:2012年14-17]
- Pentosidine, a biologically important advanced glycation endproduct, has been accessed in a rapid, high-yielding manner. The synthesis was accomplished via a six-step sequence starting with 3-amino-2-chloropyridine and f...
- Total Synthesis of Ripostatin A
[作者:TANG WUFENG; PRUSOV EVGENY V,期刊:Organic Letters, 页码:4690-4693 , 文章类型: Article,,卷期:2012年14-17]
- The first total synthesis of the bacterial RNA-polymerase inhibitor ripostatin A (1) was achieved. The route utilizes a cyclic methyl acetal intermediate and a sequence of a double Stifle cross-coupling reaction followed...
- A Pro line-Based Phosphine Template for Staudinger Ligation
[作者:PARK CHUNGMIN; NIU WEI; LIU CHUNRONG; BIGGS TYLER D; GUO JIANTAO; XIAN MING,期刊:Organic Letters, 页码:4694-4697 , 文章类型: Article,,卷期:2012年14-17]
- A proline-based phosphine template enabling a rapid Staudinger ligation of azide-containing substrates under mild conditions is reported. This reaction has a second-order rate constant of 1.12 M-1 s(-1). It is expected t...
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