- Penetratin analogues acting as antifungal agents
[作者：Garibotto, FM; Garro, AD; Rodriguez, AM; Raimondi, M; Zacchino, SA; Perczel, A; Somlai, C; Penke, B; Enriz, RD,期刊：European Journal of Medicinal Chemistry, 页码：370-377 , 文章类型： Article，,卷期：2011年46-1]
- The synthesis, in vitro evaluation, and conformational study of penetratin analogues acting as antifungal agents are reported. Different peptides structurally related with penetratin were evaluated. Analogues of penetrat...
- Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents
[作者：Chimenti, F; Bizzarri, B; Bolasco, A; Secci, D; Chimenti, P; Granese, A; Carradori, S; D'Ascenzio, M; Lilli, D; Rivanera, D,期刊：European Journal of Medicinal Chemistry, 页码：378-382 , 文章类型： Article，,卷期：2011年46-1]
- A new series of [4-(4'-substituted-phenyl)thiazol-2-yl]hydrazine derivatives were synthesized in good yield (86-99%) and characterized by elemental analysis, IR, H-1 NMR, and mass spectral studies. The compounds were ass...
- 1,2,5-Oxadiazole analogues of leflunomide and related compounds
[作者：Giorgis, M; Lolli, ML; Rolando, B; Rao, A; Tosco, P; Chaurasia, S; Marabello, D; Fruttero, R; Gasco, A,期刊：European Journal of Medicinal Chemistry, 页码：383-392 , 文章类型： Article，,卷期：2011年46-1]
- A new series of compounds, structurally related to leflunomide, based on the 1,2,5-oxadiazole ring system (furazan) has been synthesised, and their ability to undergo ring scission at physiological pH to afford the corre...
- Synthesis, biological evaluation of chrysin derivatives as potential immunosuppressive agents
[作者：Lv, PC; Cai, TT; Qian, Y; Sun, JA; Zhu, HL,期刊：European Journal of Medicinal Chemistry, 页码：393-398 , 文章类型： Article，,卷期：2011年46-1]
- A series of novel chrysin derivatives was firstly synthesized and evaluated on their immunosuppressive activity in the search for potential immunosuppressive agents. Among them, compounds 5c displayed the most potent imm...
- Synthesis and evaluation of quinonoid compounds against tumor cell lines
[作者：da Silva, EN; Cavalcanti, BC; Guimaraes, TT; Pinto, MDFR; Cabral, IO; Pessoa, C; Costa-Lotufo, LV; de Moraes, MO; de Andrade, CKZ; dos Santos, MR; de Simone, CA; Goulart, MOF; Pinto, AV,期刊：European Journal of Medicinal Chemistry, 页码：399-410 , 文章类型： Article，,卷期：2011年46-1]
- Thirty two compounds were synthesized in moderate to high yields and showed activity against cancer cells HL-60 (leukemia), MDA-MB435 (melanoma), HCT-8 (colon) and SF295 (central nervous system), with IC50 below 2 mu M f...
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