- Synthesis and biological evaluation of dehydroabietic acid derivatives
[作者:Gonzalez, MA; Perez-Guaita, D; Correa-Royero, J; Zapata, B; Agudelo, L; Mesa-Arango, A; Betancur-Galvis, L,期刊:European Journal of Medicinal Chemistry, 页码:811-816 , 文章类型: Article,,卷期:2010年45-2]
- A series of C18-oxygenated derivatives of dehydroabietic acid were synthesized from commercial abietic acid and evaluated for their cytotoxic, antimycotic, and antiviral activities. (C) 2009 Elsevier Masson SAS. All righ...
- Imidazole derivatives as possible microbicides with dual protection
[作者:Kumar, L; Sarswat, A; Lal, N; Sharma, VL; Jain, A; Kumar, R; Verma, V; Maikhuri, JP; Kumar, A; Shukla, PK; Gupta, G,期刊:European Journal of Medicinal Chemistry, 页码:817-824 , 文章类型: Article,,卷期:2010年45-2]
- Twenty seven derivatives (2-28) of 2-(2-methyl-5-nitro-1H-imidazol-1-yl)ethanol were synthesized and evaluated for anti-trichomonas, spermicidal and antifungal activities. Twenty six compounds were active against Trichom...
- Synthesis and in vitro cytostatic activity of new beta-D-arabino furan[1 ',2 ':4,5]oxazolo- and arabino-pyrimidinone derivatives
[作者:Bosc, JJ; Latxague, L; Leger, JM; Balzarini, J; Forfar, I; Jarry, C; Guillon, J,期刊:European Journal of Medicinal Chemistry, 页码:831-839 , 文章类型: Article,,卷期:2010年45-2]
- A series of nucleoside derivatives was obtained via heteroatom annulation of the amino oxazoline Of D(-)-arabinose. Unequivocal proofs for the stereostructure of some new arabinosyl pyrimidinone derivatives were obtained...
- TDAE-assisted synthesis of new imidazo[2,1-b]thiazole derivatives as anti-infectious agents
[作者:Juspin, T; Laget, M; Terme, T; Azas, N; Vanelle, P,期刊:European Journal of Medicinal Chemistry, 页码:840-845 , 文章类型: Article,,卷期:2010年45-2]
- A series of new imidazo[2,1-b]thiazoles was prepared in moderate to good yields in a four step synthesis using the TDAE methodology from 6-chloromethyl-5-nitroimidazo[2,1-b]thiazole and keto esters, ketomalonates and ket...
- Synthesis and antiviral activity of boranophosphonate isosteres of AZT and d4T monophosphates
[作者:Barral, K; Priet, S; De Michelis, C; Sire, J; Neyts, J; Balzarini, J; Canard, B; Alvarez, K,期刊:European Journal of Medicinal Chemistry, 页码:849-856 , 文章类型: Article,,卷期:2010年45-2]
- We report synthesis, in vitro antiviral activity, and stability studies in biological media of original boranophosphonate isosteres of AZT and d4T monophophates. A convenient route for the synthesis of 3'-Azido-3'-deoxyt...
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