- Unprecedented Cu(I)-Catalyzed Microwave-Assisted Three-Component Coupling of a Ketone, an Alkyne, and a Primary Amine
[作者:PERESHIVKO OLGA P; PESHKOV VSEVOLOD A; VAN DER EYCKEN ERIK V,期刊:Organic Letters, 页码:2638-2641 , 文章类型: Article,,卷期:2010年12-11]
- An efficient, microwave-assisted Cu(I)-catalyzed one-pot coupling of a ketone, an alkyne, and a primary amine (KA(2) coupling) is described, giving access to secondary propargylamines.
- Synthesis of (+/-)-Eusynstyelamide A
[作者:BARYKINA OLGA V; SNIDER BARRY B,期刊:Organic Letters, 页码:2664-2667 , 文章类型: Article,,卷期:2010年12-11]
- The synthesis of (+/-)-eusynstyelamide A has been accomplished in six steps in 13% overall yield from 6-bromoindole, methyl glycidate, and Boc-protected agmatine. If oxygen is carefully excluded from the reaction, the ke...
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