- New endomorphin analogs containing alicyclic b-amino acids: influence on bioactive conformation and pharmacology profile.
[作者:Keresztes, Attila;Szucs, Maria;Borics, Attila;Kover, Katalin E.;Forro, Eniko;Fulop, Ferenc;Tomboly, Csaba;Peter, Antal;Pahi, Annamaria;Fabian, Gabriella;Muranyi, Mariann;Toth, Geza;,期刊:Journal of Medicinal Chemistry, 页码:4270-4279 , 文章类型: 研究论文,,卷期:2008年51-14]
- Endomorphins were subjected to a no. of structural modifications in a search for their bioactive conformations. The alicyclic b-amino acids cis-(1S,2R)ACPC/ACHC, cis-(1R,2S)ACPC/ACHC, trans-(1S,2S)ACPC/ACHC, and trans-(...
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