- Synthesis of Novel Furo-, Thieno-, and Pyrroloazepines
[作者:VILLARREAL CARLOS; MARTINEZ ROBERTO,期刊:Synthesis, 页码:3346-3352 , 文章类型: Article,,卷期:2010年-19]
- The synthesis of novel furo-, thieno-, and pyrroloazepine compounds, using the oxidative radical alkylation of three five-membered heterocyclic 3-acetic acid derivatives, is described. The bicyclic systems were obtained,...
- Synthesis of 1,5,6,7-Tetrahydro-4H-pyrazolo[4,3-c]pyridin-4-ones as Conformationally Constrained Pyrazole Analogues of Histamine
[作者:ZEROVNIK DARJA; GROSELJ UROS; KRALJ DAVID; MALAVASIC CRT; BEZENSEK JURE; DAHMANN GEORG; STARE KATARINA; MEDEN ANTON; STANOVNIK BRANKO; SVETE JURIJ,期刊:Synthesis, 页码:3363-3373 , 文章类型: Article,,卷期:2010年-19]
- Three synthetic methods for the preparation of 1,5-disubstituted 1,5,6,7-tetrahydro-4H-pyrazolo[4,3-c]pyridin-4-ones as heterocyclic histamine analogues were developed. The first method starts from easily available methy...
- Synthesis of Annulated Pyrroles: Condensation of Aldose Sugars, Arylamines, and 1,3-Diones Using TBAB
[作者:NAGARAPU LINGAIAH; CHEEMALAPATI VENKATA NARASIMHAJI; KARNAKANTI SHUKLACHARY; BANTU RAJASHAKER,期刊:Synthesis, 页码:3374-3378 , 文章类型: Article,,卷期:2010年-19]
- Readily available tetrabutylammonium bromide (TBAB, 10 mol%), in the molten state, efficiently catalyzes the reaction of a variety of in situ generated enamines, from arylamines and 1,3-ketones, with aldose sugars under ...
- Synthesis of alpha-Aminocyclopropylphosphonic Acids
[作者:CHEMAGIN ANDREY V; YASHIN NIKOLAI V; GRISHIN YURI K; KUZNETSOVA TAMARA S; ZEFIROV NIKOLAI S,期刊:Synthesis, 页码:3379-3383 , 文章类型: Article,,卷期:2010年-19]
- A convenient, general approach to alpha-aminocyclopropylphosphonic acids via reduction and hydrolysis of alpha-nitrocyclopropylphosphonates is described. A number of the title compounds were synthesized in excellent yiel...
- Reactions of Substituted Oxazoles and Thiazoles with Acid Chlorides: Carbon-Carbon Bond Formation through Cyclic Ketene Acetals
[作者:CHATTERJEE SABORNIE; YE GUOZHONG; SONG YINGQUAN; BARKER BOBBY LLOYD; PITTMAN CHARLES U JR,期刊:Synthesis, 页码:3384-3394 , 文章类型: Article,,卷期:2010年-19]
- Reactions of 2,4,5-trimethyloxazole, 2,4,5-trimethylthiazole, 2-methylthiazole, and 2-ethyl-4,5-dimethylthiazole with different acid chlorides in the presence of different bases were explored. Arylvinyl esters of substit...
- Recent Advances in the Synthesis of Carbohydrate Mimetics
[作者:KOESTER DENNIS C; HOLKENBRINK ANNIKA; WERZ DANIEL B,期刊:Synthesis, 页码:3217-3242 , 文章类型: Review,,卷期:2010年-19]
- Highly diverse strategies are employed to mimic carbohydrates. Two subgroups of carbohydrate mimetics are very important: alterations of the core structure and modifications of the O-glycosidic linkage. This review prese...
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