- 5-Amino-pyrazoles as potent and selective p38 alpha inhibitors
[作者：Das, J; Moquin, RV; Dyckman, AJ; Li, TL; Pitt, S; Zhang, R; Shen, DR; McIntyre, KW; Gillooly, K; Doweyko, AM; Newitt, JA; Sack, JS; Zhang, HJ; Kiefer, SE; Kish, K; McKinnon, M; Barrish, JC; Dodd, JH; Schieven, GL; Leftheris, K,期刊：Bioorganic & Medicinal Chemistry Letters, 页码：6886-6889 , 文章类型： Article，,卷期：2010年20-S1]
- The synthesis and structure-activity relationships (SAR) of p38 alpha MAP kinase inhibitors based on a 5-amino-pyrazole scaffold are described. These studies led to the identification of compound 2j as a potent and selec...
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