- N-beta-Fmoc-N-beta-Methyl-aza-beta(3)-amino Acids
[作者:NICOLAS IRENE; KISSELJOVA KSENIJA; BAUCHAT PATRICK; BAUDYFLOCH MICHELE,期刊:SYNLETT, 页码:327-330 , 文章类型: Article,,卷期:2011年-3]
- The potential of peptides as drug candidates is limited by their poor pharmacokinetic properties. Many peptides have a short half-life, in vivo half-life, and insufficient oral availability. Inspired by the N-methylation...
- Boric Acid Mediated N-Acylation of Sulfoximines
[作者:GARIMALLAPRABHAKARAN ASWINKUMAR; HARMATA MICHAEL,期刊:SYNLETT, 页码:361-364 , 文章类型: Article,,卷期:2011年-3]
- The N-acylation of a sulfoximine with carboxylic acids was accomplished with boric acid and several boronic acids. Aliphatic acids give fair yields of products while acids related to phenylacetic and phenoxyacetic acids ...
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