- Modular Synthesis of Core Fucosylated N-Glycans
[作者:OTT DIMITRI; SEIFERT JOACHIM; PRAHL INGO; NIEMIETZ MATHAEUS; HOFFMAN JOANNA; GUDER JANNA; MOENNICH MANUEL; UNVERZAGT CARLO,期刊:European Journal of Organic Chemistry, 页码:5054-5068 , 文章类型: Article,,卷期:2012年-26]
- A modular synthesis of complex-type N-glycans containing the core fucosyl motif was optimized. The core trisaccharide building block was protected by a methoxyphenyl group for convenient core fucosylation. The trisacchar...
- Complete Characterization of the 3D Properties of the CCR5 Antagonist Vicriviroc through DFT Calculations, NMR Spectroscopy, and X-ray Analysis
[作者:LEGNANI LAURA; COLOMBO DIEGO; VILLA STEFANIA; MENEGHETTI FIORELLA; CASTELLANO CARLO; GELAIN ARIANNA; ALBINI FRANCA MARINONE; TOMA LUCIO,期刊:European Journal of Organic Chemistry, 页码:5069-5074 , 文章类型: Article,,卷期:2012年-26]
- Vicriviroc is a piperazine-based CCR5 receptor antagonist, with better oral availability, potency, safety, and pharmacological properties than those of its precursor SCH-C, but whose development has been stopped. A full ...
- Oxidative Coupling of Enolates, Enol Silanes, and Enamines: Methods and Natural Product Synthesis
[作者:GUO FENGHAI; CLIFT MICHAEL D; THOMSON REGAN J,期刊:European Journal of Organic Chemistry, 页码:4881-4896 , 文章类型: Review,,卷期:2012年-26]
- Oxidative coupling of enolates, enol silanes, and enamines provides a direct method for the construction of useful 1,4-dicarbonyl synthons. Despite its first being reported in 1935, with subsequent important advances beg...
- Total Synthesis of (+)-Seimatopolide A
[作者:REDDY CHADA RAJI; RAO NAGAVARAM NARSIMHA; REDDY MOTATIPALLY DAMODER,期刊:European Journal of Organic Chemistry, 页码:4910-4913 , 文章类型: Article,,卷期:2012年-26]
- The first enantioselective total synthesis of a polyhydroxylated macrolide, (+)-seimatopolide A, was achieved. The key reactions, Sharpless asymmetric dihydroxylation, Yamaguchi esterification, and ring-closing metathesi...
- A peri-Cyclised Naphthalene Dimer: Synthesis and Properties of an Unusual Vilsmeier-Haack Product of 1,3,6,8-Tetramethoxynaphthalene
[作者:PITTELKOW MICHAEL; NIELSEN CHRISTIAN B; BROCKNANNESTAD THEIS; SCHAUMAGNUSSEN MAGNUS; CHRISTENSEN JORN B,期刊:European Journal of Organic Chemistry, 页码:4931-4936 , 文章类型: Article,,卷期:2012年-26]
- An unusual peri-dimerised product was obtained when subjecting 1,3,6,8-tetramethoxynaphthalene to VilsmeierHaack reaction conditions (POCl3/DMF). The formation of this peri-dimerised naphthalene product suggests that 1,3...
- Synthesis of Coenzyme Q10
[作者:OH EUNTAEK; KIM HEE JIN; OH JUNG TAEK; SU LIANG; YUN INKYUN; NAM KYUNGGU; MIN JAEHONG; KIM JOON WOO; KOO SANGHO,期刊:European Journal of Organic Chemistry, 页码:4954-4962 , 文章类型: Article,,卷期:2012年-26]
- A practical synthesis of coenzyme Q10 has been developed. The route features an improved FriedelCrafts allylation of tetramethoxytoluene with a para-chlorobenzenesulfonyl-substituted C5 allylic chloride at 40 degrees C. ...
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