- Treatment Strategies of Obsessive-Compulsive Disorder and Panic Disorder/Agoraphobia
[作者:Marazziti, D; Carlini, M; Dell'Osso, L,期刊:Current Topics in Medicinal Chemistry, 页码:238-253 , 文章类型: Review,,卷期:2012年12-4]
- Anxiety disorders represent the most prevalent psychiatric disorders. In addition, a considerable burden is associated with them, not only for individual sufferers, but also for the health care system. However, many pati...
- The GABAA-BZR Complex as Target for the Development of Anxiolytic Drugs
[作者:Trincavelli, ML; Da Pozzo, E; Daniele, S; Martini, C,期刊:Current Topics in Medicinal Chemistry, 页码:254-269 , 文章类型: Review,,卷期:2012年12-4]
- Anxiety disorders have been linked to alterations in gamma-aminobutyric acid (GABA) neurotransmission. GABA interacts with the ligand-gated ion channels, GABAA receptor (GABAA-R) subtypes, and regulates the flow of chlor...
- Medicinal Chemistry of Indolylglyoxylamide GABA(A)/BzR High Affinity Ligands: Identification of Novel Anxiolytic/Non Sedative Agents
[作者:Salerno, S; Da Settimo, F; Taliani, S; Simorini, F; La Motta, C; Fornaciari, G; Marini, AM,期刊:Current Topics in Medicinal Chemistry, 页码:286-311 , 文章类型: Review,,卷期:2012年12-4]
- The classical benzodiazepines (Bz) constitute a well-known class of therapeutics displaying hypnotic, anxiolytic and anticonvulsant effects acting upon a specific binding site (BzR) belonging to the GABA(A) receptor comp...
- Geometrically Constrained Derivatives of Indolylglyoxylamides as Ligands Binding the GABA(A)/BzR Complex
[作者:Sartini, S; Morelli, M; Simorini, F; Taliani, S; Salerno, S; Marini, AM; Da Settimo, F; La Motta, C,期刊:Current Topics in Medicinal Chemistry, 页码:312-320 , 文章类型: Review,,卷期:2012年12-4]
- Indolylglyoxylamides are a class of distinctive benzodiazepine receptor ligands, proposed in the mid-eighties as open analogues of beta-carbolines. Thorough and long-lasting studies of their structure-activity relationsh...
- Medicinal Chemistry of Indolylglyoxylamide TSPO High Affinity Ligands with Anxiolytic-Like Effects
[作者:Simorini, F; Marini, AM; Taliani, S; La Motta, C; Salerno, S; Pugliesi, I; Da Settimo, F,期刊:Current Topics in Medicinal Chemistry, 页码:333-351 , 文章类型: Review,,卷期:2012年12-4]
- The mitochondrial translocator protein (TSPO) mediates the synthesis of neurosteroids in the CNS, which have been demonstrated to enhance the neurotransmitter GABA response, exhibiting related behavioural properties. Sel...
|