- Facile and Quantitative Synthesis of 1,3-Diazaheterocycle-Fused 1,2,3-Triazole Derivatives Using Fluoroalkanesulfonyl Azide as a Diazo Transfer Reagent
[作者:GU JIWEI; XIONG WANTING; ZHANG ZHENHUA; ZHU SHIZHENG,期刊:Synthesis, 页码:1717-1722 , 文章类型: Article,,卷期:2011年-11]
- A series of 1,3-diazaheterocycle-fused 1,2,3-triazoles were conveniently and quantitatively prepared by 1,3-dipolar cycloaddition of heterocyclic ketene aminals with fluoroalkanesulfonyl azide, followed by elimination of...
- A Facile Synthesis of 6H-[1,3,5]Triazino[2,1-b]quinazolin-6-ones
[作者:ABBOTT SHAUN; CLOUTIER JOSEE; HOUDE KARINE; PENNEY CHRISTOPHER; ZACHARIE BOULOS,期刊:Synthesis, 页码:1733-1740 , 文章类型: Article,,卷期:2011年-11]
- Triazinoquinazolinone derivatives are synthesized by cyclization of aminobenzamide-substituted triazine compounds in the presence of a proton source such as trifluoroacetic acid or hydrochloric acid. The reaction is mild...
- Synthesis and Biological Evaluation of Modified 2-Deoxystreptamine Dimers
[作者:COSTE GERALD; HORLACHER TIM; MOLINA LIDIA; MORENOVARGAS ANTONIO J; CARMONA ANA T; ROBINA INMACULADA; SEEBERGER PETER H; GERBERLEMAIRE SANDRINE,期刊:Synthesis, 页码:1759-1770 , 文章类型: Article,,卷期:2011年-11]
- Aminoglycosides are powerful antibiotics, but the emergence of resistant bacterial strains has prompted the search for analogues with better pharmacological profiles. The synthesis of 2-deoxystreptamine (2-DOS) dimers li...
- A New Method for the Synthesis of 1-Aryl-1,2,4-triazole Derivatives
[作者:MATIYCHUK VASYL S; POTOPNYK MYKHAYLO A; LUBORADZKI ROMAN; OBUSHAK MYKOLA D,期刊:Synthesis, 页码:1799-1803 , 文章类型: Article,,卷期:2011年-11]
- A new and convenient one-step recyclization method for the synthesis of ethyl 1-aryl-5-oxo-4,5-dihydro-1H-1,2,4-triazole-3-carboxylates is reported. Various ethyl chloro(2-arylhydrazinylidene)ethanoates react with thiazo...
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