- Regulation of CK2 by phosphorylation and O-GlcNAcylation revealed by semisynthesis
[作者:TARRANT MARY KATHERINE; RHO HEESOOL; XIE ZHI; JIANG YU LIN; GROSS CHRISTOPHER; CULHANE JEFFREY C; YAN GAI; QIAN JIANG; ICHIKAWA YOSHITAKA; MATSUOKA TATSUJI; ZACHARA NATASHA; ETZKORN FELICIA A; HART GERALD W; JEONG JUN SEOP; BLACKSHAW SETH; ZHU HENG; COLE PHILIP A,期刊:NATURE CHEMICAL BIOLOGY, 页码:262-269 , 文章类型: Article,,卷期:2012年8-3]
- Protein serine-threonine kinase casein kinase 3II (CK2) is involved in a myriad of cellular processes including cell growth and proliferation through its phosphorylation of hundreds of substrates, yet how CK2 function is...
- Menin-MLL inhibitors reverse oncogenic activity of MLL fusion proteins in leukemia
[作者:GREMBECKA JOLANTA; HE SHIHAN; SHI AIBIN; PUROHIT TRUPTA; MUNTEAN ANDREW G; SORENSON RODERICK J; SHOWALTER HOLLIS D; MURAI MARCELO J; BELCHER AMALIA M; HARTLEY THOMAS; HESS JAY L; CIERPICKI TOMASZ,期刊:NATURE CHEMICAL BIOLOGY, 页码:277-284 , 文章类型: Article,,卷期:2012年8-3]
- Translocations involving the mixed lineage leukemia (MLL) gene result in human acute leukemias with very poor prognosis. The leukemogenic activity of MLL fusion proteins is critically dependent on their direct interactio...
- Halofuginone and other febrifugine derivatives inhibit prolyl-tRNA synthetase
[作者:KELLER TRACY L; ZOCCO DAVIDE; SUNDRUD MARK S; HENDRICK MARGARET; EDENIUS MAJA; YUM JINAH; KIM YEONJIN; LEE HAKKYO; CORTESE JOSEPH F; WIRTH DYANN F; DIGNAM JOHN DAVID; RAO ANJANA; YEO CHANGYEOL; MAZITSCHEK RALPH; WHITMAN MALCOLM,期刊:NATURE CHEMICAL BIOLOGY, 页码:311-317 , 文章类型: Article,,卷期:2012年8-3]
- Febrifugine, the bioactive constituent of one of the SO fundamental herbs of traditional Chinese medicine, has been characterized for its therapeutic activity, though its molecular target has remained unknown. Febrifugin...
|