- SYNTHETIC STUDIES ON CALLIPELTINS: STEREOSELECTIVE SYNTHESES OF (3S,4R)-3,4-DIMETHYL-L-PYROGLUTAMIC ACID AND FMOC-D-ALLOTHREONINE FROM SERINE DERIVATIVES
[作者:KONNO HIROYUKI; TAKEBAYASHI YOKO; NOSAKA KAZUTO; AKAJI KENICHI,期刊:Heterocycles, 页码:79-89 , 文章类型: Article,,卷期:2010年81-1]
- The non-proteinogenic amino acids contained in callipeltins, (3S, 4R)-3, 4-dimethyl-L-pyroglutamic acid and D-allothreonine, were synthesized from D- or L-serine. The stereoselective synthesis of two methyl groups of (3S...
- SYNTHESIS OF ARNOAMINE B
[作者:NAKAHARA SHINSUKE; SADACHI TOSHIYUKI; KUBO AKINORI,期刊:Heterocycles, 页码:145-148 , 文章类型: Article,,卷期:2010年81-1]
- The synthesis of arnoamine B (2), which inhibits the catalytic activity of topoisomerase II and exhibits selective cytotoxicity against human tumor cell lines, was achieved in six steps from 5-methoxy-6-nitroindole (3) i...
- THE SYNTHESIS OF NOVEL 2,4,6-TRISUBSTITUTED 1,3,5-TRIAZINES: A SEARCH FOR POTENTIAL MURF ENZYME INHIBITORS
[作者:SOSIC IZIDOR; STEFANE BOGDAN; KOVAC ANDREJA; TURK SAMO; BLANOT DIDIER; GOBEC STANISLAV,期刊:Heterocycles, 页码:91-115 , 文章类型: Article,,卷期:2010年81-1]
- A series of new 2,4,6-trisubstituted 1,3,5-triazines, possessing a variety of substituents (-OH, -SH, -OMe, -Cl, -HNR, -SR and amino acid moieties), were synthesized and evaluated for the inhibition of the bacterial pept...
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